R715 TFA(185052-09-9 free base) ( )

Catalog No. M30810 CAS No.

COA

Datasheet

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Product Name

R715 TFA(185052-09-9 free base)
Note

Research use only, not for human use.
Brief Description

Potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Metabolically stable.
Description

Potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Metabolically stable.
Synonyms
Pathway

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Target

Other Targets
Recptor

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Research Area

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Indication

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CAS Number

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Formula Weight

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Molecular Formula

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Purity

>98% (HPLC)
Solubility

water:5 mg/mL
SMILES

CC[C@H](C)[C@H](NC(=O)[C@@H](CC1=CC2=CC=CC=C2C=C1)NC(=O)[C@H](CO)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(C)=O)C(O)=O
Chemical Name

1. Gobeil et al (1996) Structure-activity studies of B1 receptor-related peptides. Hypertension. 28 833 PMID:

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